摘要/Abstract
以不保护的单/双糖和邻氨基苯甲酰胺为原料，通过碘诱导的氧化缩合一锅法反应，合成了系列糖基喹唑啉酮衍生物，产率30%～80%，为该类化合物的合成提供了一个有效方法.碘的用量对该反应有重要的影响.
关键词: 糖基喹唑啉酮, 氧化缩合, 碘诱导
A series of aldo-quinazolinones were synthesized by a one-pot iodine-induced oxidative condensation of the unprotected mono-/di-saccharides and o-aminobenzamides in the yields of 30%~80%, providing an effective protocol for the preparation of aldo-quinazolinones. The amount of iodine has an important effect on the reaction.
Key words: aldo-quinazolinone, oxidative condensation, iodine-induced
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