摘要/Abstract
以Cu （OTf）2和AgOTf为催化剂，研究了取代邻硝基苯甲酸和取代邻氨基苯甲酰胺的选择性C-N交叉偶联反应，以中等收率合成了17个二芳基胺类苯甲酰胺.该方法为芳香胺的选择性N-芳基化提供了一种新的选择.
关键词: 脱羧反应, 选择性胺化, 邻硝基苯甲酸, 邻氨基苯甲酰胺
Cu(OTf)2/AgOTf-catalyzed selective decarboxylation C-N crossing coupling of o-nitro aromatic carboxylic acids with o-aminobenzamides has been establised, affording seventeen diarylaminobenzamides in moderate yields. The present protocol provides a new choice for selective N-arylation of amines.
Key words: decarboxylation, selective amination, o-nitro aromatic carboxylic acid, o-aminobenzamide
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