摘要/Abstract

发展了碘化亚铜催化的芳基碘化物与萘胺的分子内Ullmann类型偶联反应, 实现了萘胺分子内去芳构化芳基化反应, 以良好至优异的收率合成了一系列3H-吲哚衍生物.
关键词: Ullmann偶联, 萘胺, 芳基化, 去芳构化
A CuI-catalyzed intramolecular dearomative arylation of naphthylamines is developed through a Ullmann-type cross-coupling reaction, which led to a range of fused 3H-indole derivatives in good to excellent yields.
Key words: Ullmann coupling, naphthylamine, arylation, dearomatization


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