摘要/Abstract
通过碘介导的氧化性C-O键形成反应由易得的α，β-不饱和肟合成了一系列单、双和三取代（芳基、烷基和/或烯基）的异噁唑类化合物.该合成方法具有不使用过渡金属、操作简单、反应条件温和、反应时间短，以及底物适用范围广等优点.
关键词: 异噁唑, 碘, α,β-不饱和肟, C-O键形成
A variety of mono-, di-, and tri-substituted (aryl, alkyl, and/or alkenyl) isoxazoles were synthesized from readily accessible α,β-unsaturated oximes via I2-mediated oxidative C-O bond formation. The features of this synthetic approach include no use of transition metals, simple operation, mild reaction conditions, short reaction time, and broad substrate scope.
Key words: isoxazole, iodine, α,β-unsaturated oxime, C-O bond formation
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