摘要/Abstract

Tandem Pd(OAc)2/CuI catalyzed coupling/cyclization/chalcogenylation reaction of gem-dibromovinylanilines with boronic acids and dichalcogenides has been developed, which provides a new synthetic approach to 3-sulfenyl-and 3-selenylindoles. Various functional groups such as methoxyl, halides and trifluoromethyl groups in the substrates are tolerated.
关键词: 吲哚, Pd(OAc)2/CuI, 催化, 合成
Key words: indole, Pd(OAc)2/CuI, catalysis, synthesis
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