药学
未公开
副教授

Regioselective conversion of arenes to N-aryl-1,2,3-triazoles using C-H borylation.

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High-Throughput Discovery of Mycobacterium tuberculosis Protein Tyrosine Phosphatase B (MptpB) Inhibitors Using Click Chemist

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High-Throughput Synthesis of Azide Libraries Suitable for Direct “Click” Chemistry and in situ Screening

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Solid-phase synthesis of azidomethylene inhibitors targeting cysteine proteases

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In vivo imaging of a bacterial cell division protein using a protease-assisted small-molecule labeling approach

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Solid-phase assembly and in situ screening of protein tyrosine phosphatase inhibitors.

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"Click" synthesis of small-molecule inhibitors targeting caspases.

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Site-specific covalent labeling of proteins inside live cells using small molecule probes

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Methods of using click chemistry in the discovery of enzyme inhibitors

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Click Chemistry as a High-Throughput Amenable Platform in

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Activity-based fingerprinting of proteases.

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Rapid assembly and in situ screening of bidentate inhibitors of protein tyrosine phosphatases

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Chemical approaches for live cell bioimaging

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Expanded utility of the native chemical ligation reaction

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Cell-permeable small molecule probes for site-specific labeling of proteins