摘要/Abstract

报道了一种钯催化2-炔基芳基叠氮化合物与丙烯酸衍生物合成吲哚-3-丙烯酸酯的新方法. 该方法实现了在温和的反应条件下合成多种1H-吲哚-3-丙烯酸酯衍生物.
关键词: 钯催化, α-亚胺钯卡宾, 吲哚-3-丙烯酸酯, 丙烯酸
A novel method to prepare 1H-indol-3-yl acrylates from 2-alkynyl arylazides with acrylic acids catalyzed by Pd has been described. A variety of 1H-indol-3-yl acrylate derivatives were prepared under mild reaction conditions.
Key words: Pd-catalysis, α-imino palladium carbene, indole-3-acrylate, acrylic acid


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