删除或更新信息,请邮件至freekaoyan#163.com(#换成@)

广西民族大学化学化工学院导师教师师资介绍简介-申利群老师简况

本站小编 Free考研考试/2021-06-13



联系方式 :E-mail:liqunshen@126.com
简介:
申利群:博士,教授,硕士生导师。已主持完成国家自然科学基金1项,广西高校优秀人才资助计划1项,广西自治区自然科学基金2项,广西教育厅重点项目1项。目前主持国家自然基金(**),广西科技重大专项项目(桂科AA**)各1项,参与科技部等国家级项目3项。获教育部自然科学一等奖1项,湖南科技进步三等奖1项,邵阳市科技进步一等奖1项。先后在Angew. Chem. Int. Ed. Engl,J.Am.Chem.Soc,steroids 等国内外期刊上发表论文50多篇,获专利授权4项。长期从事药物化学、制药工艺学与药物合成反应课程教学工作。

研究领域:

1、计算机辅助药物设计合成及活性研究;
2、天然产物分离、结构修饰及活性研究


历年来获得学术成果奖情况:
1. 申利群(9/10), 教育部自然科学一等奖, 2017;
2. 申利群(2/4),湖南省科技进步奖,, 湖南省人民政府,省部级,( 三等奖 ) 排名02,2012;
3. 申利群(2/4),湖南省邵阳市科技进步一等奖,邵阳市人民政府,地厅级,( 一等奖 ) 排名02,2011。




近五年作为负责人主持科研项目情况
1、国家自然科学基金项目,**、基于Survivin蛋白靶点的甘草查尔酮B衍生物设计合成及抗肿瘤作用机理研究、2018/01-2021/12、38万元、主持。
2、广西科技重大专项项目子项目(桂科AA**)、广西药用植物沉香的产业化研究,2017/09-2020/12、30万元、主持。


近五年公开发表论文情况

1. Lingyuan Xu, Sensen Qiu, Lehe Yang, Haitang Xu, Xu Liu, Shiqian Fan, Ri Cui, Weitao Fu, Chengguang Zhao, Liqun Shen*, Liangxing Wang*, Xiaoying Huang*. Aminocyanopyridines as anti-lung cancer agents by inhibiting the STAT3 pathway Molecular Carcinogenesis. 2019; 58:1512–1525.
2. Lingyuan Xu, Lingxi Shi, Sensen Qiu, Siyu Chen, Mengsha Lin, Youqun Xiang, Chengguang Zhao, Jiandong Zhu, Liqun Shen*, Zhigui Zuo * . Design, Synthesis, And Evaluation Of Cyanopyridines As Anti-Colorectal Cancer Agents Via Inhibiting STAT3 Pathway. Drug Design, Development and Therapy, 2019:13 3369–3381.
3. 田程飘,朱伟伟,宋雅玲,牛思琪,申利群*,吴爱群*. 生姜和醋泡生姜抗菌、抗氧化和抗肿瘤活性比较研究. 食品工业科技, 2019, 14: 18-23.
4. 田程飘,宋雅玲,许海棠,牛思琪,吴志鸿,申利群*. 超临界和水蒸汽蒸馏
提取沉香精油成分分析及抗氧化、抑菌活性对比研究.中国中药杂志, 2019, 44(18): 4000-4008.
5. Ya-Ling Song, Cheng-Piao Tian, Yan Wu, Li-he Jiang, Li-Qun Shen*. Design, synthesis and antitumor activity of steroidal pyridine derivatives based on molecular docking. Steroids, 2019, 143,53–61.
6、Chao Wu , Liguang Mao , Xie Huang , Weitao Fu , Xiong Cai , Yuepiao Cai ,
Liqun Shen* , Xiaoxia Ye. Theoretical study of the intermolecular recognition mechanism between Survivin and substrate based on conserved binding mode analysis. Journal of Molecular Graphics and Modelling. 2018, 83: 53-63.
7、Wu Zhang, Qiuyu Wei, Lingling Lan, Aiqun Wu, Xiuju Yin, Liqun Shen*. Allylic oxidation of cyclic alkenes with molecular oxygen and tertbutyl hydroperoxide over copper-manganese oxides. Monatsh Chem, 2017, 148:357–365.
8、Wu Zhang, Aiqun Wu, Haitang Xua, Yuxing Mob, Jie Chen, Liqun Shen*.
Design, Synthesis, and Bioassay of Novel Compounds of Isolongifolenone Oxime Derivatives. Helv. Chim. Acta , 2016, 99, 696 – 703.
9、Wu Zhang, Dan Pan, Aiqun Wu, Liqun Shen*. Effective and mild method for converting 3β-hydroxysteroids to 3-keto steroids via DDQ/TEMPO, Steroids, 2015, 96,16–20.
10、Dan Pan,Aiqun Wu,Pengfei Li,Haitang Xu,Fuhou Lei,Liqun Shen*. Palladium-loaded renewable polymeras a green heterogeneous catalyst for cross-coupling reactions under microwave irradiation,Journal ofChemical Research.,2014, 38(12):715-718.
11、Liqun shen,yong tang,aiqun wu,dan pan,kaisheng diao,Synthesis, X-Ray Crystal Structure,andComputational Study of Novel Pyrazolo[3,4-B]pyridin-3-ol Derivatives,Phosphorus,Sulfur, and Silicon andthe Related Elements,2014,189:674-685.
12、Wu, Ai Qun,Tang, Yong,Huang, Su-Yu,Shen, Li-Qun*. Synthesis and structure of novel 6-(pyrazol-1-yl)-4-methyl-1H-pyrazolo[3,4-b]pyridine-3-ol derivatives. Research on Chemical Intermediates,2014,40(1):239-247.







相关话题/化学化工学院 广西民族大学