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西北农林科技大学化学与药学院导师教师师资介绍简介-高锦明

本站小编 Free考研考试/2021-07-07

一、个人简介
高锦明,男,教授(二级),博士生导师,陕西省教学名师,国务院政府特殊津贴专家。
1986年7月本科毕业于陕西师范大学化学专业,1998年7月硕士毕业于西北农林科技大学植物资源化学专业,2001年8月获中国科学院昆明植物研究所植物化学专业博士学位。2005年至2006年及2007年至2008年在加拿大科学院生物技术研究所做访问****和博士后。
2001年获得中国科学院院长奖学金优秀奖;先后入选教育部“优秀青年教师资助计划”、“新世纪优秀人才支持计划”。2005年获陕西省“优秀博士后”,2009年获陕西省优秀留学回国人员称号,以及2014年陕西省化学优秀工作者奖。
现任西北农林科技大学化学与药学院院长,西北农林科技大学第八、九、十、十一届学位评定委员会第十二分委会主席,西北农林科技大学第三、四届学术委员会委员。
兼任中国植物学会植物化学及资源学专业委员会委员、中国菌物学会菌物化学专业委员会副主任委员、陕西省天然产物化学生物学重点实验室主任、陕西省资源化学与可持续利用工程研究中心主任、国家自然科学基金委评审专家(会审)、陕西省高等学校教学指导委员会化生类工作委员会委员、陕西省化学会常务理事、陕西省药学会常务理事、陕西省陕南中药产业发展专家顾问。
现担任《Journal of Agricultural and Food Chemistry》、《Natural Products and Bioprospecting》、《西北农林科技大学学报(自然科学版)》及《生物质化学工程》编委。
二、科研课题
近年来,先后主持和参与国家自然科学基金、国家林业公益性行业科研专项、“十二五”国家科技支撑计划、国家重点研发计划、教育部博士学科点专项科研基金等多项国家、省部级科研项目。
三、研究领域
1、中药药效物质基础研究、天然活性成分结构改造与功能研究
2、基于靶蛋白结构的天然产物结构修饰与构效关系
3、新型小分子神经生长因子NGF类化合物发现与药物开发
4、天然产物的生物转化、生物合成与调控
四、开设课程
长期致力于有机化学、植物化学的教学与科研工作,先后承担本科生有机化学、天然药物化学等课程教学,为博、硕士研究生讲授天然产物化学进展、天然产物化学、有机分析、有机合成等课程。
五、主要教学科研成果与学术论文
近年来,申请国家发明专利40项(授权30项),获省部级一、二等奖4项,陕西省教学成果奖特等奖和二等奖各1项,主编(参编)教材、专著6部。负责主持国家级精品课程《植物化学》和国家级一流本科课程《天然产物化学》。
在Chem. Rev.、J. Am. Chem. Soc.、Nat. Prod. Rep.、Org. Lett.、Chem. Commun.、Eur. J. Med. Chem.、J. Nat. Prod.、J. Agric. Food Chem.等期刊发表SCI论文180多篇。主要论文被引4200多次,H-指数33。
代表性论文:
(1) Ling-Li Liu, Zhi-Fan Chen, Yao Liu, Dan Tang, Hua-Hua Gao, Qiang Zhang, and Jin-Ming Gao*. Molecular networking-based the target discovery of potent antiproliferative polycyclic macrolactam ansamycins from Streptomyces cacaoi subsp. asoensis . Organic Chemistry Frontiers , 2020, doi: 10.1039/D0QO00557F.
(2) Xia Yin,Thi M. L. Tuong, Jun-Mian Tian, Gennaro Pescitelli*, Jin-Ming Gao*. Ganorbifates A and B from Ganoderma orbiforme, Determined by DFT Calculations of NMR data and ECD spectra, Chem. Commun. 2020, 56, 10195-10198. doi: 10.1039/D0CC04679E.
(3) Zhai, Yi-Jie; Huo, Guang-Ming; Zhang, Qiang; Li, Ding; Wang, Da-Cheng; Qi, Jian-Zhao; Han, Wen-Bo*; Jin-Ming Gao.* Phaeosphaones: tyrosinase inhibitory thiodiketopiperazines from an endophytic Phaeosphaeria fuckelii , J. Nat. Prod. 2020, 83(5), 1592–1597. http://dx.doi.org/10.1021/acs.jnatprod.0c00046.
(4) Wen-Bo Han,Guang-Yi Wang, Jiang-Jiang Tang, Wen-Ji Wang,Han Liu, Roberto R. Gil, Armando Navarro-Vázquez, Xinxiang Lei,* Jin-Ming Gao*. Herpotrichones A and B, two intermolecular [4+2] adducts with anti-neuroin?ammatory activity from a Herpotrichia species. Org. Lett. 2020, 22(2), 405–409. http://dx.doi.org/10.1021/acs.orglett.9b04099.
(5) Hong Yin, Wen-Jia Dan, Bo-Yi Fan, Chao Guo,Kui Wu, Kui-Feng Xian, Gennaro Pescitelli,* Jin-Ming Gao*. Anti-inflammatory and α -glucosidase inhibitory activities of labdane and norlabdane diterpenoids from the rhizomes of Amomum villosum , J. Nat. Prod. 2019, 82(11), 2963–2971. doi: 10.1021/acs.jnatprod.9b00283.
(6) Tang, Dan; Xu, Yuanzhen; Wang, Weiwei; Yang, Zhi; Liu, Bo; Stadler, Marc; Liu, Lingli*; Gao, Jin-Ming*. Cyathane Diterpenes From Cultures of the Bird’s Nest Fungus Cyathus hookeri and Their Neurotrophic and Anti-neuroinflammatory Activities. J. Nat. Prod. 2019, 82(6),1599-1608. doi: 10.1021/acs.jnatprod.9b00091.
(7) Wen-Jia Dan, Qiang Zhang, Fan Zhang, Wei-Wei Wang & Jin-Ming Gao*, Benzonate derivatives of acetophenone as potent α-glucosidase inhibitors: synthesis, structure-activity relationship, and mechanism. Journal of Enzyme Inhibition and Medicinal Chemistry , 2019, 34(1): 937-945. doi: 10.1080/**.2019.**.
(8) Xi-Tao Yan, Zhen An, Dan Tang, Guang-Rui Peng, Chen-Yu Cao, Yuan-Zhen Xu, Chun-Huan Li, Pei-Liang Liu, Zai-Min Jiang, Jin-Ming Gao*. Polycyclic polyprenylated acylphloroglucinol and phenolic metabolites from the aerial parts of Hypericum elatoides and their neuroprotective and anti-neuroinflammatory activities. Phytochemistry 2019, 159, 65-74. doi: 10.1016/j.phytochem.2018.12.011.
(9) Yu-Bin Bai, Zaigang Luo, Yuguang Wang, Jin-Ming Gao*, Liming Zhang*. Au-Catalyzed Intermolecular [2+2] Cycloadditions between Chloroalkynes and Unactivated Alkenes. J. Am. Chem. Soc. 2018, 140: 5860–5865. doi: 10.1021/jacs.8b01813.
(10) Dan Tang, Ling-Li Liu,Qiu-Rui He, Wen Yan, Ding Li, Jin-Ming Gao*. Ansamycins with potential anti-proliferative and anti-neuroinflammatory activity from the moss soil-derived Streptomyces cacaoi subsp. asoensis H2S5. J. Nat. Prod. 2018, 81(9):1984-1991. doi: 10.1021/acs.jnatprod.8b00203.
(11) Chen-Yu Cao, Cheng-Chen Zhang, Xin-Wei Shi, Ding Li, Wei Cao, Xia Yin, Jin-Ming Gao*, Sarcodonin G derivatives exhibit distinctive effects on neurite outgrowth by modulating NGF signaling in PC12 Cells, ACS Chem. Neurosci. 2018, 9, 1607–1615. doi: 10.1021/acschemneuro.7b00488.
(12) Jing Wei, Yuanyuan Cheng, Wan-Hui Guo, Da-Cheng Wang, Qiang Zhang, Ding Li, Jianhui Rong*, Jin-Ming Gao*. Molecular diversity and potential anti-neuroinflammatory activities of cyathane diterpenoids from the Basidiomycete Cyathus africanus. Scientific Reports , 2017, 7: 8883. doi: 10.1038/s41598-017-09118-z.
(13) Qiang Zhang, Hao-Yu Tang, Min Chen,Jie Yu, Hui Li, Jin-Ming Gao*. Natural products driven diversity via skeletal remodeling of caryophyllene β-lactam. Org. Biomol. Chem. 2017, 15(20): 4456-4463. doi: 10.1039/c7ob00741h.
(14) Xin Yu, Jiadong Hu, Zhigao Shen, Hui Zhang, Jin-Ming Gao, Weiqing Xie*. Stereospecific construction of contiguous quaternary all-carbon centers by oxidative ring contraction. Angew. Chem. I nt. Ed. Engl. 2017, 56(1): 350–353. doi: 10.1002/anie..
(15) Shuai Dong, Kiran Indukuri, Derrick L. J. Clive*, Jin-Ming Gao*. Models of the BC ring systems of MPC1001 and MPC1001F. Chem. Commun. 2016, 52, 8271-8274. doi: 10.1039/c6cc04169h.
(16) Bo Luo, Jin-Ming Gao*, Mark Lautens*. Palladium-catalyzed norbornene-mediated tandem amination/cyanation reaction: a new method for the convergent synthesis of ortho -aminated benzonitriles. Org. Lett. 2016, 18, 4166?4169.
(17) Bai, Rui; Zhang, Cheng-Chen; Yin, Xia; Wei, Jing; Gao, Jin-Ming*. Cyathane diterpenoids with neurotrophic activity from cultures of the fungus Cyathus striatus . J. Nat. Prod. 2015, 78(4): 783–788. doi: 10.1021/np501030r.
(18) Bai, Meng-Meng; Shi, Wei; Tian, Jun-Mian; Lei Ming; Kim, Young Ho; Kim, Jang Hoon*; Sun, Ya Nan; Gao, Jin-Ming*. Soluble epoxide hydrolase inhibitory and anti-inflammatory components from the leaves of Eucommia ulmoides Oliver (Duzhong). J. Agri. Food Chem. 2015 , 63 (8): 2198–2205. doi: 10.1021/acs.jafc.5b00055.
(19) Shuai Dong, Jiang-Jiang Tang*, Cheng-Chen Zhang, Jun-Mian Tian, Jun-Tao Guo, Qiang Zhang, He Li, Jin-Ming Gao*.Semisynthesis and in vitr o cytotoxic evaluation of new analogues of 1- O -acetylbritannilactone, a sesquiterpene from Inula britannica . Eur. J. Med. Chem. 2014, 80 , 71–82. doi: 10.1016/j.ejmech.2014.04.028.
(20) Jin-Ming Gao*, Sheng-Xiang Yang, Jian-Chun Qin. Azaphilones: Chemistry and Biology, Chemical Reviews , 2013, 113(7): 4755–4811. doi: 10.1021/cr300402y.
六、联系方式
通讯地址:陕西杨凌西农路22号 西北农林科技大学化学与药学院
邮编:712100
电话: 邮箱:jinminggao@nwsuaf.edu.cn



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